Magnetic Yeast Glucan Particles for Antibody-Free Separation of Viable Macrophages from <i>Drosophila melanogaster</i>

✅ 全文

磁性酵母葡聚糖颗粒用于从黑腹果蝇中无抗体分离活巨噬细胞

作者 Gabriela Krejčová; Ivan Saloň; Vojtěch Klimša; Pavel Ulbrich; Ayse Beyza Aysan; Adam Bajgar; František Štĕpánek 期刊 ACS Biomaterials Science & Engineering 发表日期 2023 ISSN 2373-9878 DOI 10.1021/acsbiomaterials.3c01199 类型 原创研究 (Original Research)

📄 英文摘要 English Abstract

EN

Currently available methods for cell separation are generally based on fluorescent labeling using either endogenously expressed fluorescent markers or the binding of antibodies or antibody mimetics to surface antigenic epitopes. However, such modification of the target cells represents potential contamination by non-native proteins, which may affect further cell response and be outright undesirable in applications, such as cell expansion for diagnostic or therapeutic applications, including immunotherapy. We present a label- and antibody-free method for separating macrophages from living Drosophila based on their ability to preferentially phagocytose whole yeast glucan particles (GPs). Using a novel deswelling entrapment approach based on spray drying, we have successfully fabricated yeast glucan particles with the previously unachievable content of magnetic iron oxide nanoparticles while retaining their surface features responsible for phagocytosis. We demonstrate that magnetic yeast glucan particles enable macrophage separation at comparable yields to fluorescence-activated cell sorting without compromising their viability or affecting their normal function and gene expression. The use of magnetic yeast glucan particles is broadly applicable to situations where viable macrophages separated from living organisms are subsequently used for analyses, such as gene expression, metabolomics, proteomics, single-cell transcriptomics, or enzymatic activity analysis.

📄 中文摘要 Chinese Abstract

中文
目前可用的细胞分离方法通常基于荧光标记,利用内源性表达的荧光标记物或抗体/抗体模拟物与表面抗原表位的结合。然而,这种对靶细胞的修饰引入了非天然蛋白的潜在污染,可能影响细胞的后续反应,并且在某些应用中完全不可取,例如用于诊断或治疗用途(包括免疫治疗)的细胞扩增。 酵母全葡聚糖颗粒(GPs)是由β-葡聚糖为主形成的多孔多糖壳,通过一系列洗涤和提取步骤从常见的酿酒酵母中获得。尽管原始酵母的大部分细胞成分已被去除,GPs仍保留表面结构特征,使其能被免疫细胞表面的dectin-1受体识别并被主动吞噬。GPs的这一特性已在离体和体内得到充分证实。 最近研究表明,注射到活体果蝇体内的GPs迅速分布于血淋巴中,并被巨噬细胞选择性摄取,且不影响其正常功能。GPs的这一特性可用于通过磁场实现无标记巨噬细胞分离,但迄今为止,科学界尚未在保持GPs形态和表面分子基团不受影响的前提下实现足够高的磁响应。

📋 英文结构化总结 English Structured Summary

全文整理

EN

Header:

Background

Currently available methods for cell separation are generally based on fluorescent labeling using either endogenously expressed fluorescent markers or the binding of antibodies or antibody mimetics to surface antigenic epitopes. However, such modification of the target cells represents potential contamination by non-native proteins, which may affect further cell response and be outright undesirable in applications, such as cell expansion for diagnostic or therapeutic applications, including immunotherapy.

Whole yeast glucan particles (GPs) are porous polysaccharide shells predominantly formed by β-glucans, obtained from common baker’s yeast by a series of washing and extraction steps. Although most cellular components of the original yeast are removed, GPs retain surface structural features that make them readily recognized by dectin-1 receptors of immune cells and actively phagocytosed. This property of GPs has been well documented both ex vivo and in vivo.

It has been recently shown that GPs injected into living Drosophila are rapidly distributed through the hemolymph and selectively taken up by macrophages without compromising their normal function. This feature of GPs could be used for label-free macrophage separation by a magnetic field, but achieving sufficiently high magnetic response of GPs without compromising their morphology and surface molecular motifs has so far eluded the scientific community.

Header:

Methods

Preparation of Yeast Glucan Particles GPs were obtained from baker’s yeast (Saccharomyces cerevisiae) using a series of washing and extraction steps as reported previously. 25 g portion of baker’s yeast was added into 100 mL of 1 M NaOH and mixed to form a suspension, and the material was heated for 1 h at 90 °C and then centrifuged at 14,500 g for 5 min (Dynamica Velocity 14, Austria). The supernatant was discarded, and this step was repeated twice. The processed alkali-insoluble solids were

Header:

Results

We have successfully fabricated yeast glucan particles with the previously unachievable content of magnetic iron oxide nanoparticles while retaining their surface features responsible for phagocytosis.

We demonstrate that magnetic yeast glucan particles enable macrophage separation at comparable yields to fluorescence-activated cell sorting without compromising their viability or affecting their normal function and gene expression.

We report a comprehensive physicochemical characterization of magnetic GPs and demonstrate their in vivo biodistribution, cell uptake, and successful application for magnetic separation.

Header:

Data Summary

No quantitative results or key statistics are provided in the extracted text.

Header:

Conclusions

The use of magnetic yeast glucan particles is broadly applicable to situations where viable macrophages separated from living organisms are subsequently used for analyses, such as gene expression, metabolomics, proteomics, single-cell transcriptomics, or enzymatic activity analysis.

Header:

Practical Significance

The use of magnetic yeast glucan particles is broadly applicable to situations where viable macrophages separated from living organisms are subsequently used for analyses, such as gene expression, metabolomics, proteomics, single-cell transcriptomics, or enzymatic activity analysis. This label- and antibody-free method avoids contamination by non-native proteins, which is particularly important for diagnostic or therapeutic applications including immunotherapy.

📋 中文结构化总结 Chinese Structured Summary

中文

背景:

目前可用的细胞分离方法通常基于荧光标记,利用内源性表达的荧光标记物或抗体/抗体模拟物与表面抗原表位的结合。然而,这种对靶细胞的修饰引入了非天然蛋白的潜在污染,可能影响细胞的后续反应,并且在某些应用中完全不可取,例如用于诊断或治疗用途(包括免疫治疗)的细胞扩增。

酵母全葡聚糖颗粒(GPs)是由β-葡聚糖为主形成的多孔多糖壳,通过一系列洗涤和提取步骤从常见的酿酒酵母中获得。尽管原始酵母的大部分细胞成分已被去除,GPs仍保留表面结构特征,使其能被免疫细胞表面的dectin-1受体识别并被主动吞噬。GPs的这一特性已在离体和体内得到充分证实。

最近研究表明,注射到活体果蝇体内的GPs迅速分布于血淋巴中,并被巨噬细胞选择性摄取,且不影响其正常功能。GPs的这一特性可用于通过磁场实现无标记巨噬细胞分离,但迄今为止,科学界尚未在保持GPs形态和表面分子基团不受影响的前提下实现足够高的磁响应。

方法:

酵母葡聚糖颗粒的制备:按照先前报道的方法,从酿酒酵母(Saccharomyces cerevisiae)中通过一系列洗涤和提取步骤获得GPs。将25 g酿酒酵母加入100 mL 1 M NaOH中混合形成悬浮液,将材料在90 °C加热1小时,然后在14,500 g下离心5分钟(Dynamica Velocity 14,奥地利)。弃去上清液,此步骤重复两次。处理后的碱不溶性固体被

结果:

我们成功制备了含有此前无法实现的高含量磁性氧化铁纳米颗粒的酵母葡聚糖颗粒,同时保留了负责吞噬作用的表面特征。

我们证明磁性酵母葡聚糖颗粒能够以与荧光激活细胞分选相当的产量实现巨噬细胞分离,且不影响其活力或正常功能和基因表达。

我们报告了磁性GPs的全面理化表征,并证明了其在体内的生物分布、细胞摄取以及磁分离的成功应用。

数据摘要:

提取的文本中未提供定量结果或关键统计数据。

结论:

磁性酵母葡聚糖颗粒广泛适用于从活体生物中分离存活巨噬细胞并随后用于分析的场景,例如基因表达、代谢组学、蛋白质组学、单细胞转录组学或酶活性分析。

实际意义:

磁性酵母葡聚糖颗粒广泛适用于从活体生物中分离存活巨噬细胞并随后用于分析的场景,例如基因表达、代谢组学、蛋白质组学、单细胞转录组学或酶活性分析。这种无标记、无抗体的方法避免了非天然蛋白的污染,这对于包括免疫治疗在内的诊断或治疗应用尤为重要。

📖 英文全文 English Full Text

EN

pmc ACS Biomater Sci Eng ACS Biomater Sci Eng 822 acssd ab ACS Biomaterials Science & Engineering 2373-9878 pmc-is-collection-domain yes pmc-collection-title ACS AuthorChoice PMC10777351 PMC10777351.1 10777351 10777351 38048070 10.1021/acsbiomaterials.3c01199 1 Article Magnetic

Yeast Glucan Particles for Antibody-Free Separation of Viable Macrophages from Drosophila melanogaster Krejčová Gabriela † Saloň Ivan ‡ Klimša Vojtěch ‡ Ulbrich Pavel § Aysan Ayse Beyza ‡ Bajgar Adam * † ‡ https://orcid.org/0000-0001-9288-4568 Štěpánek František * ‡ † Department of Molecular Biology and Genetics, Faculty of Sciences, University of South Bohemia , Branišovská 1160/31, 37005 České Budějovice, Czech Republic ‡ Department of Chemical Engineering, University of Chemistry and Technology Prague , Technická 5, 166 28 Prague 6, Czech Republic § Department of Biochemistry and Microbiology, University of Chemistry and Technology , Prague, Technická 5, 166 28 Prague 6, Czech Republic * Email: bajgaa00@prf.jcu.cz . * Email: stepanef@vscht.cz . 04 12 2023 08 01 2024 10 1 453061 355 364 22 08 2023 16 11 2023 02 11 2023 10 01 2024 11 01 2024 09 09 2024 © 2023 The Authors. Published by American Chemical Society 2023 The Authors https://creativecommons.org/licenses/by/4.0/ Permits the broadest form of re-use including for commercial purposes, provided that author attribution and integrity are maintained ( https://creativecommons.org/licenses/by/4.0/ ). Currently available methods for cell separation are generally based on fluorescent labeling using either endogenously expressed fluorescent markers or the binding of antibodies or antibody mimetics to surface antigenic epitopes. However, such modification of the target cells represents potential contamination by non-native proteins, which may affect further cell response and be outright undesirable in applications, such as cell expansion for diagnostic or therapeutic applications, including immunotherapy. We present a label- and antibody-free method for separating macrophages from living Drosophila based on their ability to preferentially phagocytose whole yeast glucan particles (GPs). Using a novel deswelling entrapment approach based on spray drying, we have successfully fabricated yeast glucan particles with the previously unachievable content of magnetic iron oxide nanoparticles while retaining their surface features responsible for phagocytosis. We demonstrate that magnetic yeast glucan particles enable macrophage separation at comparable yields to fluorescence-activated cell sorting without compromising their viability or affecting their normal function and gene expression. The use of magnetic yeast glucan particles is broadly applicable to situations where viable macrophages separated from living organisms are subsequently used for analyses, such as gene expression, metabolomics, proteomics, single-cell transcriptomics, or enzymatic activity analysis. β-glucan particles iron oxide nanoparticles spray drying cell separation phagocytosis Grantová Agentura Ceské Republiky 10.13039/501100001824 19-26127X Grantová Agentura Ceské Republiky 10.13039/501100001824 20-14030S pmc-status-qastatus 0 pmc-status-live yes pmc-status-embargo no pmc-status-released yes pmc-prop-open-access yes pmc-prop-olf no pmc-prop-manuscript no pmc-prop-legally-suppressed no pmc-prop-has-pdf yes pmc-prop-has-supplement yes pmc-prop-pdf-only no pmc-prop-suppress-copyright no pmc-prop-is-real-version no pmc-prop-is-scanned-article no pmc-prop-preprint no pmc-prop-in-epmc yes pmc-license-ref CC BY document-id-old-9 ab3c01199 document-id-new-14 ab3c01199 ccc-price Introduction Cell manipulation and processing are crucial operations in biomedical research when working with living animals, tissues, and cells. Doing it in a lean and effective manner without compromising cellular functions is key to the further use of separated cells. Currently used techniques include micro pipetting, 1 microfluidics, 2 high-gradient magnetic cell sorting, 3 and predominantly fluorescence-activated cell sorting (FACS). 4 Existing methods are generally based on fluorescent labeling of the target cells using either endogenously expressed fluorescent markers or the binding of antibodies or antibody mimetics to surface antigenic epitopes. In the case of magnetic cell sorting, the currently used methods use antigen-coupled magnetic nanoparticles that bind to the cell surface. While these approaches are perfectly acceptable in many applications such as ex post metabolomic analysis, there are also situations where the addition of non-native proteins to the separated cells is undesirable, 5 , 6 particularly if the cells are to be used for immuno-analysis and diagnostic or therapeutic purposes. 7 The cell viability can be compromised, and normal cellular functions including immune response can be affected by phenomena such as antigen shedding. 8 From the regulatory perspective in cell therapy, the contamination of the therapeutic product by nonautologous or adventitious proteins can be problematic. Whole yeast glucan particles (GPs) are porous polysaccharide shells predominantly formed by β-glucans, obtained from common baker’s yeast by a series of washing and extraction steps. 9 Although most cellular components of the original yeast are removed, GPs retain surface structural features that make them readily recognized by dectin-1 receptors of immune cells and actively phagocytosed. This property of GPs has been well documented both ex vivo 10 , 11 and in vivo. 12 , 13 Owing to their immunogenicity and porous nature, GPs lend themselves as vehicles for the encapsulation and targeted delivery of various bioactive substances. 14 − 17 Proposed diagnostic and therapeutic applications of GPs include their use as vaccine adjuvants, 18 as immuno-active drug delivery systems for the treatment of inflammatory bowel disease, as a means of improving the bioavailability of poorly soluble drugs via lymphatic transport, 13 or as contrast agents for imaging. 19 , 20 It has been recently shown that

GPs injected into living Drosophila are rapidly distributed through the hemolymph and selectively taken up by macrophages without compromising their normal function. 9 This feature of GPs could be used for label-free macrophage separation by a magnetic field, but achieving sufficiently high magnetic response of GPs without compromising their morphology and surface molecular motifs has so far eluded the scientific community. In the present work, we introduce a novel method that yields composite GPs with an unprecedentedly strong response to magnetic field while retaining their structural and functional properties. The method is based on encapsulating independently prepared magnetic iron oxide nanoparticles (IONs) into GPs by spray drying. A solvent temporarily swells the polysaccharide GP shell, enabling colloidally stable magnetic IONs to diffuse into the inner structure. By rapid solvent evaporation during spray drying, the polysaccharide shell deswells and magnetic nanoparticles are irreversibly trapped within the GPs at a high concentration, while a native GP surface is preserved. We report a comprehensive physicochemical characterization of magnetic GPs and demonstrate their in vivo biodistribution, cell uptake, and successful application for magnetic separation. Furthermore, we show that the normal function and gene expression profiles of the separated macrophages are preserved. Materials and Methods Preparation of Yeast Glucan

Particles GPs were obtained from baker’s yeast ( Saccharomyces cerevisiae ) using a series of washing and extraction steps as reported previously. 14 25 g portion of baker’s yeast was added into 100 mL of 1 M NaOH and mixed to form a suspension, and the material was heated for 1 h at 90 °C and then centrifuged at 14,500 g for 5 min (Dynamica Velocity 14, Austria). The supernatant was discarded, and this step was repeated twice. The processed alkali-insoluble solids were then mixed with 10 mL of HCl solution (pH 4.5), heated to 75

°C for 2 h, and then centrifuged at 14,500 g for 5 min. The insoluble solids were washed 3 times in deionized water, 4 times in isopropanol, and finally 2 times in acetone. Each washing step was followed by centrifugation at 14,500 g for 5 min. The final product was freeze-dried to form a white dry powder and stored in a refrigerator for further use. Preparation of Yeast GPs Modified with Rhodamine B As a reference for visualization experiments, Rhodamine B-modified yeast GPs (GP-RhodB) were prepared by dispersing 50 mg of glucan particles in 10 mL of 0.1 M carbonate-bicarbonate buffer with pH 9.2 containing

1 mg of Rhodamine B isothiocyanate dissolved in 500 μL of ethanol in a round-bottom flask. The suspension was sonicated in a sonication bath for 15 min. The suspension was then kept at 37 °C for 12 h under constant magnetic stirring at 500 rpm. The content of the reaction mixture was then washed 16 times and centrifuged for 3 min at 6000 g. The supernatant-containing unreacted material was discarded, and the obtained pellet was freeze-dried and stored in a refrigerator for further use. Synthesis of Dextran-Coated Iron Oxide Nanoparticles Dextran-coated IONs were synthesized as follows: 0.75 g of iron(III) chloride hexahydrate (Sigma-Aldrich) and 0.375 g of iron(II) chloride tetrahydrate (Sigma-Aldrich) were dissolved in 15 mL of deionized water and kept in a 100 mL three-neck flask equipped with a reverse cooler in a nitrogen atmosphere under vigorous stirring. 500 mg of

70 kDa dextran (Sigma-Aldrich) dissolved in 25 mL of deionized water was added, the mixture was then heated to 85 °C, and 2.5 mL of

25% NH 4 OH (Penta) was added dropwise into the reaction vessel. The reaction mixture was kept at 85 °C for 1 h and then cooled to room temperature. The nanoparticles were separated by magnetic decantation and washed 3 times with deionized water. The nanoparticle suspension was subsequently dialyzed for 24 h against deionized water.

The dialysate was sonicated for 10 min in a sonication bath and centrifuged at 1500 g for 5 min to remove any larger agglomerates. After centrifugation, the supernatant was filtered by a 0.2 μm PVDF (polyvinylidene difluoride) filter to obtain a nanoparticle suspension. 21 , 22 Preparation of Magnetic Yeast Glucan Particles Composite magnetic yeast GPs (mGPs) containing dextran-coated IONs were prepared by spray drying, as shown schematically in Figure 1 . 100 mg of yeast GPs (either plain GPs or

GP-RhodB) was dispersed and homogenized by ULTRA-TURRAX in a prepared mixture containing 500 μL of IONs (0.215 mg/mL), 25 mL of deionized water, and 75 mL of 96% ethanol. After dispersing, the suspension was immediately spray-dried using a Mini Spray Dryer B-290 (Büchi,

Switzerland) operated in an inert loop under a N 2 atmosphere.

Spray drying was conducted using a 1.4 mm diameter, a 2-fluid nozzle, and operating conditions consisting of 120 °C inlet temperature,

5 mL/min suspension feed rate, and 800 L/h (50%) N 2 flow rate. 15 The outlet temperature was 70–75

°C. Figure 1 Scheme of the mGP preparation process by spray drying. Left: overall process scheme. Right: mechanism of IONs embedding into GPs during droplet evaporation in the spray drying chamber. Particle Size Analysis The size distribution of the prepared magnetic nanoparticles (IONs) was evaluated by dynamic light scattering (DLS), using a Zetasizer Nano-ZS (Malvern Instruments,

UK). Before the measurement, 10 μL of the sample was added to

2 mL of deionized water, filtered by a 0.2 μm PVD filter, and placed into a disposable cuvette. The size distribution of GPs, mGPs, and mGPs-RhodB was evaluated by the static light scattering method using the Horiba Partica LA 950/S2 instrument. Prior to the measurement, the particle suspension was sonicated by Sonopuls HD 3100 (Bandelin

Electronic) for 5 min at 25 W without pulses. Electron Microscopy The surface morphology and shape of GPs and mGPs were examined by a scanning electron microscope Jeol

JCM- 5700. Samples were sputter-coated (Emitech K550X) with a 5 nm layer of gold prior to scanning electron microscopy (SEM) analysis.

Transmission electron microscopy (TEM) Jeol JEM-1010 was used for the examination of the size and surface morphology of IONs and mGPs, without any staining procedure prior to the analyses. The elemental analysis of mGPs was determined by energy-dispersive X-ray spectroscopy (EDX) using the Thermo Scientific Phenom ProX desktop SEM with Phenom

EDS software and semiautomated scanning option. Atomic Absorption

Spectroscopy The iron content in mGP samples and in solution was evaluated by atomic absorption spectroscopy (AAS) using Agilent 280FS AA with a flame atomization technique. The

Fe (Flame) method at 248.3 nm was used with a flame type: acetylene–air. X-ray Powder Diffraction Tthe crystallinity and the presence of iron oxide in composite mGPs were evaluated by recording the diffraction intensities of the samples from 6° to 110°

2θ angle using a PANaytical X’Pert PRO with a High Score

Plus diffractometer. Data evaluation was performed in the software package HighScore Plus 4.0. Drosophila melanogaster Strains and Culture The flies were raised on a standard diet containing cornmeal (80 g/L), sucrose (50 g/L), yeast (40 g/L), agar (10.433 g/L), and 10% methylparaben (16.7 mL/L) and were maintained in a humidity-controlled environment with a natural 12 h/12 h light/dark cycle at 25 °C.

We used CrqGal4 > GFP fly line for the visualization of macrophages.

This strain carries a macrophage-specific driver Crq Gal4 and reporter gene (enhanced green fluorescent protein eGFP) under the control of artificial UAS promoter (genotype w 1118 / w 1118 ; Crq-Gal4, UAS-2xeGFP/Crq-Gal4, UAS-2xeGFP ). Injection of Flies The suspension of IONs, mGPs, or mGPs-RhodB was prepared by sonication on an ice bath for 5 min at

25 W and vortexed just before injection to ensure well-dispersed particles.

CrqGal4 > GFP male flies were anaesthetized using CO 2 and injected with 50 nL of 0.1% (w/w) suspension, in case of mGPs or mGPs-RhodB, into the ventrolateral side of the abdomen using an Eppendorf Femtojet microinjector. Visualization of Magnetic Yeast GPs'

Distribution In Vivo To analyze magnetic particle distribution in Drosophila , CrqGal4 > GFP flies were injected with 50 nL of 0.1% (w/w) mGPs or mGPs-RhodB. After 45 min, the fly abdomens were opened in 4% PFA (Polysciences) in PBS and fixed for 20 min. Subsequently, the tissues were washed in PBS. Aqua Polymount (Polysciences) was used to mount the sample. The samples were imaged using an inverted fluorescent microscope (Olympus IX71) or a confocal microscope (Olympus FluoView

1000). Visualization of mGPs Uptake by Drosophila Phagocytes To visualize mGPs' uptake by Drosophila -phagocytosing cells, we prepared samples for confocal and both SEM and TEM. For the analysis using a confocal microscope, CrqGal4 > GFP flies were injected with 50 nL of 0.1% (w/w) mGPs-RhodB. After 45 min, the fly abdomens were opened in a drop of PBS on an imaging slide in order to wash up the macrophages, which were let to attach to the imaging slide for 25 min. Subsequently, the macrophages were fixed with 4%

PFA (Polysciences) in PBS. After 20 mi, the samples were stained with

Alexa Fluor Plus 405 Phalloidin (Invitrogen) for 40 min. Aqua Polymount (Polysciences) was used to mount the sample. Macrophages were imaged using an Olympus FluoView 3000 confocal microscope. For the

SEM analysis, CrqGal4 > GFP flies were injected with 50 nL of 0.1% (w/w) mGPs. After 45 min, the fly abdomens were opened in PBS and fixed in 2.5% glutaraldehyde in 0.1 M phosphate buffer (pH = 7.2) for 1 week at 4 °C. Subsequently, the opened abdomens were dehydrated through an acetone series and dried to critical point by point dryer

CPD 2 (Pelco TM) and attached to an aluminum target. For contrasting, the samples were coated with gold by using a sputter-coated E5100 (Polar Equipment Ltd.). Macrophages were examined with JEOL SEM JSM

7401F. Electron images were false colorized in Adobe Photoshop software. For the TEM analysis, CrqGal4 > GFP flies were injected with

50 nL of 0.1% (w/w) mGPs. After 45 min, the fly abdomens were cut off and placed in 2.5% glutaraldehyde in 0.1 M phosphate buffer (pH =

7.2) for 1 week at 4 °C. Subsequently, the samples for TEM were postfixed in osmium tetroxide for 2 h at 4 °C, washed at 4 °C, dehydrated through an acetone serie, and embedded in EPON resin. A series of ultrathin sections were prepared by using a Leica UCT ultramicrotome (Leica Microsystems), counterstained with uranyl acetate and lead citrate, and subsequently examined in a JEOL TEM 1010 operated at

80 kV. The TEM images were false colorized in Adobe Photoshop software. Magnetic Yeast GPs' Separation of Macrophages At 60 min after injection of mGPs, the flies were washed in PBS and homogenized in 600 mL of PBS using a pestle. The homogenate was sieved through a nylon strainer (40 μm). This strainer was then additionally washed with 200 μL of PBS, which was subsequently added to the homogenate subsequently. The samples were centrifuged (3 min, 4 °C,

3500 rpm), and the supernatant was washed with ice-cold PBS after each centrifugation (3 times). Prior to mGPs separation, samples were transferred to FACS polystyrene tubes by using a disposable bacterial filter (50 μm, Sysmex). The macrophages were separated from the sample using the QuadroMACS Separator (Miltenyi Biotec) according to the manufacturer′s protocol. In brief, the magnetic LS column (Miltenyi Biotec) was placed in the QuadroMACS Separator and rinsed before isolation with equilibrative buffer (PBS, 0.5% BSA, 2 mM EDTA, pH 7.2). Subsequently, the sample with the cell suspension was loaded into the LS column, and the flow through was discarded. To wash off the remaining cells, the LS column was washed 3 times with 1 mL of equilibrative buffer (Miltenyi Biotec). To obtain the phagocytosing cells, the LS column was removed from the QuadroMACS Separator and washed with 2 mL of rinsing buffer (PBS, 0.5% BSA, 2 mM EDTA, pH 7.2), and the flow though was collected into a nuclease free Eppendorf tube. Analysis of Macrophage Viability after Magnetic Separation The macrophages obtained by mGPs' separation were allowed to attach to the imaging slide for 25 min. Subsequently, the macrophages were fixed with 4% paraformaldehyde (PFA) in PBS (Polysciences). After

20 min, the samples were stained with Alexa Fluor Plus 405 Phalloidin (Invitrogen) for 40 min. Aqua polymount (Polysciences) was used to mount the sample. The macrophages were imaged using an Olympus FluoView

3000 confocal microscope. Apart from visual assessment of cytoskeleton remodeling, cell viability was also determined quantitatively by letting the isolated macrophages spread on the surface of the Neubauer counting chamber, staining by trypan blue in a ratio of 1:1 to a final concentration of 0.02%, and counting. FACS Isolation of Macrophages As a reference experiment, the GFP-expressing macrophages were isolated from CrqGal4 > GFP male flies using fluorescence-activated cell sorting (FACS). Three hundred flies were anesthetized with CO 2 , washed in PBS, and homogenized in 600 mL of PBS using a pestle. The homogenate was sieved through a nylon cell strainer (40 μm). This strainer was then additionally washed with 200 μL of PBS, which was added to the homogenate subsequently. The samples were centrifuged (3 min, 4 °C, 800 g ), and the supernatant was washed with ice-cold PBS after each centrifugation (3 times). Prior to sorting, samples were transferred to FACS polystyrene tubes using a disposable bacterial filter (50 μm, Sysmex), and macrophages were sorted into 100 μL of

PBS using a S3TM Cell Sorter (BioRad). Isolated cells were verified by fluorescence microscopy and differential interference contrast. Gene Expression Analysis Gene expression analysis was performed on 100 000 isolated macrophages. The macrophages were isolated by a cell sorter (S3e Cell Sorter, BioRad) as described in the section

Isolation of Macrophages, transferred to TRIzol Reagent (Invitrogen), and homogenized using a DEPC-treated pestle. Subsequently, RNA was extracted with TRIzol Reagent (Invitrogen) according to the manufacturer’s protocol. Superscript III Reverse Transcriptase (Invitrogen) primed by an oligo(dT)20 primer was used for reverse transcription. Relative expression rates for particular genes were quantified on a CFX 1000

Touch Real-Time Cycler (BioRad) using the TP 2× SYBR Master Mix (Top-Bio) in three technical replicates with the following protocol: initial denaturation −3 min at 95 °C, amplification −15 s at 94 °C, 20 s at 56 °C, and 25 s at 72 °C for 40 cycles. Melting curve analysis was performed at 65–85 °C/step

0.5 °C. The qPCR data were analyzed using double delta Ct analysis, and the expressions or specific genes were normalized to the expression of Ribosomal protein 49 (Rp49) in the corresponding sample. The relative values (fold change) to the control are shown in the graphs. Samples for gene expression analysis were collected from three independent experiments. Primer Sequences Rp49 forward: AAGCTGTCGCACAAATGGCG 30 , 31 Rp49 reverse: GCACGTTGTGCACCAGGAAC Hemolectin forward: GCGTACGAAGGAGATTCTC Hemolectin reverse: CACCTCGTGCTTCTGTGT Croquemort forward: CTTCTGGCCGGGTATTGCAG Croquemort reverse: GCTTTCATAGGCATCAGT Lactate dehydrogenase forward: CAGAGAAGTGGAACGAGCTG Lactate dehydrogenase reverse: CATGTTCGCCCAAAACGGAG Basket forward: TACGGCCCATAGGATCAGGT Basket reverse: CCCTATATGCTCGCTTGGCA Relish forward: ACAGGACCGCATATCG Relish reverse: GTGGGGTATTTCCGGC Diptericin A forward: GCTGCGCAATCGCTTCTACT Diptericin A reverse: TGGTGGAGTGGGCTTCATG Defensin forward: GTTCTTCGTTCTCGTGG Defensin reverse: CTTTGAACCCCTTGGC Metchnikowin forward: AACTTAATCTTGGAGCGA Metchnikowin reverse: CGGTCTTGGTTGGTTAG Drosocin forward: CCATCGTTTTCCTGCT Drosocin reverse: CCATCGTTTTCCTGCT Enolase forward: CAACATCCAGTCCAACAAGG Enolase reverse: GTTCTTGAAGTCCAGATCGT Phosphofructosekinase forward: AGCTCACATTTCCAAACATCG Phosphofructosekinase reverse: TTTGATCACCAGAATCACTGC Phosphoglucose isomerase forward: ACTGTCAATCTGTCTGTCCA Phosphoglucose isomerase reverse: GATAACAGGAGCATTCTTCTCG Unpaired3 forward: AGAACACCTGCAATCTGAAGC Unpaired3 reverse: TCTTGGTGCTCACTGTGGCC Imaginal morphogenesis protein late 2 forward: TTCGCGGTTTCTGGGCACCC Imaginal morphogenesis protein late 2 reverse: GCGCGTCCGATCGTCGCATA Eiger forward: AGCTGATCCCCCTGGTTTTG Eiger reverse: GCCAGATCGTTAGTGCGAGA Stat92E forward: CTGGGCATTCACAACAATCCAC Stat92E reverse: GTATTGCGCGTAACGAACCG. Results and Discussion Physicochemical Properties of mGPs After the incorporation of IONs by spray drying, mGPs retained the characteristic wrinkled ellipsoid shape known from plain GPs ( Figure 2 a,b). The volume-mean particle size of mGPs determined by laser diffraction was 5.1 ± 1.9 μm ( Figure 2 c), which is consistent both with the size of original yeast and with the values previously reported for unmodified GPs. 14 The fact that the incorporation of magnetic particles did not cause aggregation or changes in the surface morphology of mGPs is crucial for subsequent uptake by phagocytosing cells. Energy-dispersive X-ray spectroscopy (EDX) of plain and mGPs ( Figure 2 d,e) proved the presence of IONs in mGPs. The Fe content of mGPs determined by EDX was 1.4% ( Table 1 ). The iron content determined independently by AAS was 1.2 ± 0.1%. TEM analysis revealed that IONs were uniformly distributed within the polysaccharide shell of mGPs ( Figure 2 f). Prior to their incorporation into mGPs, dextran-coated IONs had a volume-mean diameter of 124.1 nm (measured by DLS in water) with a polydispersity index of 0.144 ( Figure 2 g inset).

After incorporation into mGPs, IONs remained well dispersed within the glucan shell ( Figure 2 g). Note that the individual iron oxide cores visible as darker spots in the TEM image are smaller than the equivalent hydrodynamic diameter of fully hydrated dextran-coated IONs measured by DLS. This is because the dextran coating is not distinguishable from the beta-glucan background and also because magnetic nanoparticles are known to form temporary clusters in aqueous media. Table 1 EDX Analysis of mGPs sample element symbol atomic number atomic concentration % plain GPs C 6 81.7 O 8 18.3 Fe 26 0.0 mGPs C 6 76.9 O 8 21.7 Fe 26 1.4 Figure 2 (a) SEM of plain glucan particles. (b) SEM of mGPs. The scale bars in both SEMs are 8 μm. (c) Particle size distribution of mGPs in water, measured by static light scattering; the volume-mean particle size is 5.1 ± 1.9 μm. (d) EDX spectrum of plain GPs. (e)

EDX spectrum of mGPs, proving the presence of iron. The macroscopic manifestation of the presence of iron oxide in mGPs is their attraction to a magnet as shown in the inset. (f) TEM of a single mGP. The scale bar represents 1000 nm. (g) Detailed TEM showing how IONs are entrapped and uniformly dispersed within the mGP shell. The scale bar represents

200 nm. The volume-weighted particle size distribution of dextran-coated

IONs in water before incorporation into mGPs, measured by DLS, is shown as inset. (h) XRPD spectra of IONs, plain GPs, and mGPS, proving the presence of iron oxide in mGPs. The presence of iron oxide in the composite mGPs was additionally proven by measuring the XRPD spectra ( Figure 2 h). The characteristic crystalline peaks of iron oxide at 21.5°, 35.1°, 67.3°, and 74.4°

2θ were clearly visible in mGPs, while no such peaks were present in plain GPs. A crucial feature with respect to further application is the stability of mGPs in aqueous media in terms of ION retention.

To detect potential loss of IONs during magnetic manipulation in an aqueous medium, mGPs were repeatedly separated by a magnet and redispersed.

No free IONs could be detected in the supernatant, indicating that the embedding of IONs in the polysaccharide shell of mGPs was sufficiently strong to prevent the loss of magnetic properties over time. The full characterization of the magnetic properties of IONs including magnetization curves at 5 and 300 K and field-cooled and zero-field-cooled susceptibility have been reported in our recent work. 29 The macroscopic manifestation of their magnetic properties is the ability to attract mGPs to a permanent magnet and separate them from solution, as shown in Figure 2 . Biodistribution and Macrophage Uptake of mGPs For investigating the biodistribution of mGPs and subsequent magnetic separation of viable macrophages, a Drosophila melanogaster strain bearing an endogenous construct for GFP protein expression in macrophages (Crq > Gal4; UAS2xGFP) was employed. Such macrophages are easily recognized for assaying their morphology and counting.

The injection of 0.1% w/w mGPs led to a fast systemic distribution through the opened circulatory system of the fly ( Figure 3 a). Within 20–30 min after injection, mGPs could be found throughout the body of adult Drosophila including the distal parts. Within 1 h after injection, clear colocalization in areas occupied by macrophages was observable ( Figure 3 b), which is consistent with the in vivo behavior of plain GPs reported earlier. The internalization of mGPs by macrophages has been proven by the analysis of whole-body cross sections by SEM and TEM ( Figure 3 c–e). Analysis of dissected immune cells revealed that macrophages internalized multiple mGPs ( Figure 3 f). In a control experiment, free IONs (not encapsulated in mGPs) injected into adult flies were found not to specifically accumulate in macrophages ( Figure S1 , Supporting Information). Figure 3 (a) Time progress of mGP biodistribution in Drosophila after injection.

Within 20 min, mGPs reach even distal parts of the body of adult flies. (b) Distribution of mGPs (red) in adult Drosophila at 1 h after injection, showing colocalization with macrophages (green). (c) Pseudocolored SEM micrograph showing the process of engulfment of mGPs (red) by a macrophage (green) at

20 min after injection. (d) Pseudocolored TEM micrograph showing the localization of endocytosed mGPs (red) in the macrophages (green) at 1 h after injection. (e) TEM micrograph showing the detail of an endocytosed mGP (red) in the cytosol of the Drosophila macrophage (green). (f) Representative confocal image of a phagocytosing cell (green) from a CrqGal4 > GFP adult Drosophila injected by mGPs (red) at 1 h after injection. Actin was stained by phalloidin (cyan). Magnetic Cell Separation and Gene Expression Flies injected with mGPs were homogenized 45 min after particle administration, and the homogenates were used for magnetic column separation (QuadroMACS

Separator, LS Columns, Miltenyi Biotec). In parallel, tissue homogenates from flies injected only with a buffer were processed by FACS separation of GFP-expressing macrophages as a control ( Figure 4 a). The statistical data accompanying Figure 4 a based on four independent biological replicas are summarized in Table 2 . Before magnetic separation, the homogenate contained 0.458% ± 0.049% of GFP-positive cells (macrophages).

The residue after magnetic separation contained 0.042% ± 0.006% of GFP-positive cells, which represents approximately 9.3% of the original. Thus, magnetic separation was able to extract approximately

90.7% of all GFP-positive cells originally present in the homogenate, which is comparable to the yield obtained from FACS. The sensitivity of the method, defined as the fraction of macrophages targeted by mGP administration, was 97.9% ± 2.5% ( N = 90;

4 replicates), while its selectivity, defined as the fraction macrophages within the population of cells that have engulfed mGPs, was 100% ±

0% ( N = 100; 5 replicates). Details of the sensitivity and selectivity measurements are provided in Supporting Information . The subsequent isolation of RNA from samples obtained by both approaches provided a comparable amount of RNA ( Figure 4 d). This was confirmed by quantifying purified RNA on a nanodrop instrument and quantifying the expression level of Rp49, commonly used as a housekeeping gene in Drosophila . The concentration of Rp49 in the case of macrophages separated by mGPs and by FACS was 630.6 ± 117.3 and 586.9 ± 115.4 ng/μL, respectively. Table 2 Sort Data Accompanying Figure 4 a before mag. separation Rep.1 Rep.2 Rep.3 Rep.4 average st. dev. sorted cells 10,123,021 10,185,447 10,066,524 10,121,254 10,124,062 48,606 GFP positive 43,528 52,561 48,211 41,231 46,383 5040 percent 0.430 0.516 0.479 0.407 0.458 0.049 after mag. separation Rep.1 Rep.2 Rep.3 Rep.4 average st. dev. sorted cells 10,185,894 10,024,653 10,144,874 10,132,241 10,121,916 68,768 GFP positive 4086 5112 3844 4117 4290 562 percent 0.040 0.051 0.038 0.041 0.042 0.006 Figure 4 (a) Schematic representation of the cell separation process. Upper panel: CrqGal4 > GFP adult flies were injected with 50 nL of 0.1% (w/w) mGPs. The flies were homogenized, and the homogenate was magnetically sieved, resulting in the retention of approximately 90% of phagocytosing cells. The permeate was collected and FACS sorted based on the endogenously expressed GFP signal (G2 gate). The sorter detected the residual 10% of unseparated macrophages, constituting 0.04% out of the overall cell count. Lower panel: In a reference macrophage isolation experiment without mGP injection, the macrophages were sorted from the homogenate only by FACS, giving a yield of 0.46% out of the overall cell count ( Table 2 ). The phagocytosing cells obtained by mGPs-based magnetic separation and FACS sorter show comparable viability and were subsequently used for RT-qPCR. (b) Visualization of the injection of adult fly with mGPs. (c) Confocal microscopy visualization of croquemort and phalloidin present in living macrophages after magnetic separation. (d) Quantification of the expression level of Rp49 (commonly used as a housekeeping gene in Drosophila ) for magnetically and FACS-sorted macrophages. The viability of the magnetically separated macrophages determined by the tryptophan blue assay was 95.5%. The good condition of the isolated cells manifested itself also by their characteristic spreading phenotype on the surface of a microscopic slide and cytoskeleton remodeling ( Figure 4 c). Finally, the expression level of macrophage-specific markers (hemolectin, croquemort), immune-related genes (defensin, drosocin, metchnikowin, diptericin

A), and characteristic readout of cellular stress pathways (Relish, basket) were analyzed for both techniques, revealing that macrophages separated by means of magnetic glucan particles possess natural physiological features ( Figure 5 ).

This indicates that the mGP were not cytotoxic and their uptake did not cause any anomalous physiological response in the macrophages.

The expression level of inflammatory cytokines was not found to be significantly different between magnetically separated and FACS-sorted macrophages ( Figure 5 ), indicating that neither the engulfment of mGPs nor the magnetic separation process itself resulted in the activation of the inflammatory response. The macrophages separated by means of mGPs can in principle be subsequently used for various analyses such as gene expression analysis, metabolomics, proteomics, single-cell transcriptomics, and enzymatic activity analysis. 7 , 23 − 25 Figure 5 Comparison of gene expression of macrophage markers (croquemort, hemolectin), glycolytic gene (lactate dehydrogenase, enolase, phosphofructokinase, phosphoglucose isomerase), stress and immune response genes (basket,

Relish, STAT92e), antimicrobial peptides (metchnikowin, diptericin

A, drosocin, defensin), and cytokines (Eiger, Upd2, Upd3, ImpL2) in phagocytosing cells obtained by mGPs-based magnetic separation and

FACS sorter. The results were compared by two-way ANOVA followed by

Tukey’s multiple comparison test. Expression levels normalized against Rp49 are reported as fold change relative to the levels of the analyzed gene expression in mGPs-separated phagocytes, which were arbitrarily set to 1. The individual dots represent biological replicates with line/bar showing mean ± SD, asterisks mark statistically significant differences (* p < 0.05; ** p < 0.01), and NS marks statistically insignificant differences. Conclusions We have prepared mGPs using a new approach based on the deswelling of porous polysaccharide shell during rapid solvent evaporation during spray drying. This enables the irreversible entrapment of a large quantity of independently prepared IONs into the mGP structure, in which they remain homogeneously dispersed without undesired agglomeration of clustering. When injected into living Drosophila , mGP quickly spread across the body and were readily and selectively taken up by macrophages. This enabled subsequent macrophage isolation from tissue homogenates by a magnetic separation column. 26 − 28 The key to the successful application of mGPs for magnetic cell separation were three properties: (i) preservation of the size, surface morphology and structural motifs characteristic of original GPs, which are a prerequisite for immune recognition and efficient phaogcytosis; (ii) high concentration of embedded IONs, which is a prerequisite for generating a sufficiently strong response of the particles to an external magnetic field; and (iii) biocompatibility, which is prerequisite for good viability and further application of the isolated cells without compromising normal cellular functions and gene expression. Unlike magnetic separation based on attaching magnetic beads to the external cell surface via specific antibodies, the method based on mGPs has several advantages: (i) it enables antibody- and label-free isolation of immune cells; (ii) it covers all cells in the host organism that may participate in the engulfment of pathogens, with no need for knowing these cells a priori; (iii) due to a highly evolutionarily conserved feature (phagocytosis), the method can be used basically in all animals, not just insects; and (iv) the method allows short processing time, it is gentle, and the cells are exposed only to physiological buffers and no additional chemicals. Overall, it can be concluded that the fabrication of magnetic yeast GPs (mGPs) represents a suitable strategy for isolating macrophages, sufficient in amount and quality to perform gene expression analyses. Since this approach is independent of having endogenously expressed fluorescent markers or binding of cells via specific antibodies against the surface antigenic epitope, it may also be adapted for other situations where it is desirable to separate a population of live phagocytic cells from insect and noninsect species. Of course, it should also be noted that the presence of mGPs in the macrophages may not be universally desirable (e.g., when studying iron metabolism), but based on the data presented in this work (viability, functionality, and gene expression), the magnetically separated macrophages were not negatively affected by the engulfment of mGPs. Supporting Information Available The Supporting

Information is available free of charge at https://pubs.acs.org/doi/10.1021/acsbiomaterials.3c01199 . Results of a reference experiment in which free IONs (i.e., not embedded within mGPs) were injected into Drosophila ; information on the evaluation of selectivity, sensitivity, and purity of the magnetic separation method; and information about the gating strategy used for cell sorting ( PDF ) Supplementary Material ab3c01199_si_001.pdf Author Contributions G.K. and I.S. have contributed equally to this work. I.S., G.K., A.B., and F.Š. conceived the project. I.S., G.K., and V.K. conducted the experiments.

A.B.A. developed a method for the preparation of nanoparticles and synthesized IONs. P.U. analyzed nanoparticles and composite particles on TEM. I.S., G.K., A.B., and F.Š. designed the experiments and analyzed the results. A.B. and F.Š. supervised the study, provided guidance, and funding. I.S., G.K., A.B., and F.Š. wrote the initial draft of the manuscript. I.S. and F.Š. wrote the final manuscript with input from all authors. The authors declare no competing financial interest. Acknowledgments We would like to acknowledge financial support by the Czech Science Foundation, project nos. 19-26127X (F.S.) and 20-14030S (A.B.). References Hochmuth R. M.

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# 磁性酵母葡聚糖颗粒用于从黑腹果蝇中无抗体分离活体巨噬细胞

## 摘要

目前可用的细胞分离方法通常基于荧光标记,利用内源性表达的荧光标记物或抗体/抗体模拟物与表面抗原表位的结合。然而,这种对靶细胞的修饰代表了非天然蛋白的潜在污染,可能影响细胞的进一步反应,并且在某些应用中(如用于诊断或治疗目的的细胞扩增,包括免疫治疗)是完全不可取的。我们提出了一种无需标记和抗体的方法,基于巨噬细胞优先吞噬完整酵母葡聚糖颗粒(GPs)的能力,从活体果蝇中分离巨噬细胞。采用一种基于喷雾干燥的新型溶胀-包埋方法,我们成功制备了含有此前无法实现的高含量磁性氧化铁纳米颗粒的酵母葡聚糖颗粒,同时保留了其负责吞噬作用的表面特征。我们证明,磁性酵母葡聚糖颗粒能够以与荧光活化细胞分选相当的产率实现巨噬细胞分离,且不影响其活力或正常功能和基因表达。磁性酵母葡聚糖颗粒的使用广泛适用于从活体生物中分离活体巨噬细胞并随后用于基因表达、代谢组学、蛋白质组学、单细胞转录组学或酶活性分析等研究的场景。

## 引言

细胞操作和处理是生物医学研究中处理活体动物、组织和细胞时的关键操作。在不损害细胞功能的情况下以精简高效的方式进行处理,是分离细胞进一步使用的关键技术。目前使用的技术包括微量移液、微流体、高梯度磁细胞分选,以及最主要的荧光活化细胞分选(FACS)。现有方法通常基于使用内源性表达的荧光标记物或抗体/抗体模拟物与表面抗原表位的结合来对靶细胞进行荧光标记。在磁细胞分选的情况下,目前使用的方法采用与抗原偶联的磁性纳米颗粒与细胞表面结合。虽然这些方法在许多应用中(如事后代谢组学分析)完全可以接受,但在某些情况下,向分离的细胞中添加非天然蛋白是不可取的,特别是当细胞用于免疫分析和诊断或治疗目的时。细胞活力可能受到损害,包括免疫反应在内的正常细胞功能可能受到抗原脱落等现象的影响。从细胞治疗监管的角度来看,治疗产品被非自体或外来蛋白的污染可能存在问题。

完整酵母葡聚糖颗粒(GPs)是由β-葡聚糖主要形成的多孔多糖壳,通过一系列洗涤和提取步骤从普通面包酵母中获得。尽管原始酵母的大部分细胞成分被去除,但GPs保留了使其能够被免疫细胞表面的dectin-1受体识别并主动吞噬的表面结构特征。GPs的这一特性已在离体和体内得到充分记录。由于其免疫原性和多孔性质,GPs适合作为各种生物活性物质的封装和靶向递送载体。GPs的拟议诊断和治疗应用包括用作疫苗佐剂、用于治疗炎症性肠病的免疫活性药物递送系统、通过淋巴转运改善难溶性药物的生物利用度,或用作成像的对比剂。最近的研究表明,注射到活体果蝇中的GPs通过血淋巴快速分布,并被巨噬细胞选择性摄取,且不影响其正常功能。GPs的这一特性可用于通过磁场实现无标记的巨噬细胞分离,但迄今为止,在不损害GPs形态和表面分子基团的前提下实现足够高的磁性响应一直是科学界面临的挑战。

在本工作中,我们介绍了一种新方法,该方法制备的复合GPs具有前所未有的强磁场响应,同时保持其结构和功能特性。该方法基于通过喷雾干燥将独立制备的磁性氧化铁纳米颗粒(IONs)包封到GPs中。溶剂使多糖GP壳暂时溶胀,使胶体稳定的磁性IONs扩散到内部结构中。通过喷雾干燥过程中的快速溶剂蒸发,多糖壳发生退溶胀,磁性纳米颗粒以不可逆的方式高浓度截留在GPs内,同时保留了天然的GP表面。我们报道了磁性GPs的综合物理化学表征,并证明了其在体内的生物分布、细胞摄取以及磁性分离的成功应用。此外,我们表明分离的巨噬细胞的正常功能和基因表达谱得以保留。

## 材料与方法

### 酵母葡聚糖颗粒的制备

如前所述,从面包酵母(酿酒酵母)中通过一系列洗涤和提取步骤获得GPs。将25克面包酵母加入100毫升1 M NaOH中混合形成悬浮液,将材料在90°C加热1小时,然后以14,500 g离心5分钟(Dynamica Velocity 14,奥地利)。弃去上清液,重复此步骤两次。然后将处理后的碱不溶性固体与10 mL HCl溶液(pH 4.5)混合,在75°C加热2小时,然后以14,500 g离心5分钟。将不溶性固体用去离子水洗涤3次,用异丙醇洗涤4次,最后用丙酮洗涤2次。每次洗涤步骤后均以14,500 g离心5分钟。将最终产物冷冻干燥形成白色干粉,储存在冰箱中备用。

### 罗丹明B修饰酵母GPs的制备

作为可视化实验的参考,通过将50 mg葡聚糖颗粒分散在10 mL pH 9.2的0.1 M碳酸盐-碳酸氢盐缓冲液(含1 mg罗丹明B异硫氰酸酯溶于500 μL乙醇中)中,在圆底烧瓶中制备罗丹明B修饰的酵母GPs(GP-RhodB)。将悬浮液在超声浴中超声处理15分钟。然后将悬浮液在37°C下以500 rpm恒速磁力搅拌保持12小时。然后将反应混合物的内容物洗涤16次并以6000 g离心3分钟。弃去含有未反应材料的上清液,将所得沉淀冷冻干燥并储存在冰箱中备用。

### 葡聚糖包覆氧化铁纳米颗粒的合成

葡聚糖包覆IONs的合成如下:将0.75 g六水合氯化铁(III)(Sigma-Aldrich)和0.375 g四水合氯化铁(II)(Sigma-Aldrich)溶解在15 mL去离子水中,在氮气氛围下置于装有回流冷凝器的100 mL三颈烧瓶中,剧烈搅拌。加入500 mg 70 kDa葡聚糖(Sigma-Aldrich)溶于25 mL去离子水的溶液,将混合物加热至85°C,然后将2.5 mL 25% NH4OH(Penta)逐滴加入反应容器中。将反应混合物在85°C保持1小时,然后冷却至室温。通过磁性倾析分离纳米颗粒,并用去离子水洗涤3次。随后将纳米颗粒悬浮液对去离子水透析24小时。将透析液在超声浴中超声处理10分钟,并以1500 g离心5分钟以去除任何较大的团聚体。离心后,通过0.2 μm PVDF(聚偏二氟乙烯)过滤器过滤上清液以获得纳米颗粒悬浮液。

### 磁性酵母葡聚糖颗粒的制备

含有葡聚糖包覆IONs的复合磁性酵母GPs(mGPs)通过喷雾干燥制备,如图1所示。将100 mg酵母GPs(普通GPs或GP-RhodB)分散并通过ULTRA-TURRAX在含有500 μL IONs(0.215 mg/mL)、25 mL去离子水和75 mL 96%乙醇的制备混合物中均质化。分散后,使用Mini Spray Dryer B-290(Büchi,瑞士)在N2氛围下以惰性回路操作立即进行喷雾干燥。喷雾干燥使用1.4 mm直径的双流体喷嘴进行,操作条件包括120°C入口温度、5 mL/min悬浮液进料速率和800 L/h(50%)N2流速。出口温度为70–75°C。

**图1** 通过喷雾干燥制备mGP过程的示意图。左:整体过程示意图。右:在喷雾干燥室中液滴蒸发期间IONs嵌入GPs的机制。

### 粒径分析

使用Zetasizer Nano-ZS(Malvern Instruments,英国)通过动态光散射(DLS)评估制备的磁性纳米颗粒(IONs)的粒径分布。测量前,将10 μL样品加入2 mL经0.2 μm PVD过滤器过滤的去离子水中,放入一次性比色皿中。使用Horiba Partica LA 950/S2仪器通过静态光散射法评估GPs、mGPs和mGPs-RhodB的粒径分布。测量前,将颗粒悬浮液通过Sonopuls HD 3100(Bandelin Electronic)以25 W超声处理5分钟,不使用脉冲。

### 电子显微镜

使用扫描电子显微镜Jeol JCM-5700检查GPs和mGPs的表面形态和形状。样品在扫描电子显微镜(SEM)分析前通过溅射镀膜(Emitech K550X)镀上5 nm金层。透射电子显微镜(TEM)Jeol JEM-1010用于检查IONs和mGPs的尺寸和表面形态,分析前不使用任何染色程序。mGPs的元素分析通过能量色散X射线光谱(EDX)使用Thermo Scientific Phenom ProX台式SEM配合Phenom EDS软件和半自动扫描选项确定。

### 原子吸收光谱

使用Agilent 280FS AA配合火焰原子化技术通过原子吸收光谱(AAS)评估mGP样品和溶液中的铁含量。使用248.3 nm处的Fe(火焰)方法,火焰类型:乙炔-空气。

### X射线粉末衍射

通过记录样品在6°至110° 2θ角范围内的衍射强度,使用PANaytical X'Pert PRO配合High Score Plus衍射仪评估复合mGPs的结晶度和氧化铁的存在。在HighScore Plus 4.0软件包中进行数据评估。

### 黑腹果蝇品系和培养

果蝇在含有玉米粉(80 g/L)、蔗糖(50 g/L)、酵母(40 g/L)、琼脂(10.433 g/L)和10%对羟基苯甲酸甲酯(16.7 mL/L)的标准饮食上饲养,并在25°C、自然12小时/12小时光/暗循环的湿度控制环境中维持。我们使用CrqGal4 > GFP果蝇品系进行巨噬细胞可视化。该品系携带巨噬细胞特异性驱动子Crq Gal4和在人工UAS启动子控制下的报告基因(增强绿色荧光蛋白eGFP)(基因型w1118/w1118;Crq-Gal4, UAS-2xeGFP/Crq-Gal4, UAS-2xeGFP)。

### 果蝇注射

将IONs、mGPs或mGPs-RhodB的悬浮液在冰浴上以25 W超声处理5分钟制备,注射前涡旋以确保颗粒良好分散。将CrqGal4 > GFP雄性果蝇用CO2麻醉,使用Eppendorf Femtojet显微注射器向腹部外侧注射50 nL 0.1%(w/w)悬浮液(对于mGPs或mGPs-RhodB)。

### 磁性酵母GPs体内分布的可视化

为了分析果蝇中磁性颗粒的分布,向CrqGal4 > GFP果蝇注射50 nL 0.1%(w/w)mGPs或mGPs-RhodB。45分钟后,在PBS中的4% PFA(Polysciences)中打开果蝇腹部并固定20分钟。随后,将组织在PBS中洗涤。使用Aqua Polymount(Polysciences)封片样品。使用倒置荧光显微镜(Olympus IX71)或共聚焦显微镜(Olympus FluoView 1000)对样品成像。

### mGPs被果噬细胞摄取的可视化

为了可视化mGPs被果蝇吞噬细胞的摄取,我们制备了用于共聚焦以及SEM和TEM分析的样品。对于使用共聚焦显微镜的分析,向CrqGal4 > GFP果蝇注射50 nL 0.1%(w/w)mGPs-RhodB。45分钟后,在成像载玻片上的PBS液滴中打开果蝇腹部以洗涤巨噬细胞,使其附着在成像载玻片上25分钟。随后,用PBS中的4% PFA(Polysciences)固定巨噬细胞。20分钟后,将样品用Alexa Fluor Plus 405 Phalloidin(Invitrogen)染色40分钟。使用Aqua Polymount(Polysciences)封片样品。使用Olympus FluoView 3000共聚焦显微镜对巨噬细胞成像。

对于SEM分析,向CrqGal4 > GFP果蝇注射50 nL 0.1%(w/w)mGPs。45分钟后,在PBS中打开果蝇腹部,在0.1 M磷酸盐缓冲液(pH = 7.2)中的2.5%戊二醛中于4°C固定1周。随后,将打开的腹部通过丙酮系列脱水,并通过临界点干燥器CPD 2(Pelco TM)干燥,并连接到铝靶上。为了对比,使用溅射镀膜E5100(Polar Equipment Ltd.)用金涂覆样品。使用JEOL SEM JSM 7401F检查巨噬细胞。在Adobe Photoshop软件中对电子图像进行伪彩色处理。

对于TEM分析,向CrqGal4 > GFP果蝇注射50 nL 0.1%(w/w)mGPs。45分钟后,切下果蝇腹部,置于0.1 M磷酸盐缓冲液(pH = 7.2)中的2.5%戊二醛中于4°C固定1周。随后,TEM样品在四氧化锇中于4°C后固定2小时,在4°C洗涤,通过丙酮系列脱水,并包埋在EPON树脂中。使用Leica UCT超薄切片机(Leica Microsystems)制备一系列超薄切片,用乙酸铀酰和柠檬酸铅反染色,然后在80 kV下操作的JEOL TEM 1010中检查。在Adobe Photoshop软件中对TEM图像进行伪彩色处理。

### 磁性酵母GPs分离巨噬细胞

注射mGPs后60分钟,将果蝇在PBS中洗涤,并用研杵在600 mL PBS中均质化。将匀浆通过尼龙过滤器(40 μm)过滤。然后用200 μL PBS额外洗涤该过滤器,随后将其加入匀浆中。将样品离心(3分钟,4°C,3500 rpm),每次离心后用冰冷的PBS洗涤上清液(3次)。在mGPs分离之前,使用一次性细菌过滤器(50 μm,Sysmex)将样品转移到FACS聚苯乙烯管中。使用QuadroMACS分离器(Miltenyi Biotec)根据制造商的方案从样品中分离巨噬细胞。简言之,将磁性LS柱(Miltenyi Biotec)放入QuadroMACS分离器中,在分离前用平衡缓冲液(PBS、0.5% BSA、2 mM EDTA、pH 7.2)冲洗。随后,将含有细胞悬浮液的样品加载到LS柱中,弃去流穿液。为了洗涤剩余的细胞,用1 mL平衡缓冲液(Miltenyi Biotec)洗涤LS柱3次。为了获得吞噬细胞,将LS柱从QuadroMACS分离器中取出,用2 mL冲洗缓冲液(PBS、0.5% BSA、2 mM EDTA、pH 7.2)洗涤,将流穿液收集到无核酸酶的Eppendorf管中。

### 磁性分离后巨噬细胞活力的分析

将通过mGPs分离获得的巨噬细胞附着在成像载玻片上25分钟。随后,用PBS中的4%多聚甲醛(PFA)固定巨噬细胞。20分钟后,将样品用Alexa Fluor Plus 405 Phalloidin(Invitrogen)染色40分钟。使用Aqua polymount(Polysciences)封片样品。使用Olympus FluoView 3000共聚焦显微镜对巨噬细胞成像。除了细胞骨架重塑的视觉评估外,还通过让分离的巨噬细胞在Neubauer计数室表面铺展,以1:1比例用台盼蓝染色至终浓度0.02%,然后计数来定量确定细胞活力。

### FACS分离巨噬细胞

作为参考实验,使用荧光活化细胞分选(FACS)从CrqGal4 > GFP雄性果蝇中分离表达GFP的巨噬细胞。将三百只果蝇用CO2麻醉,在PBS中洗涤,并用研杵在600 mL PBS中均质化。将匀浆通过尼龙细胞过滤器(40 μm)过滤。然后用200 μL PBS额外洗涤该过滤器,随后将其加入匀浆中。将样品离心(3分钟,4°C,800 g),每次离心后用冰冷的PBS洗涤上清液(3次)。分选前,使用一次性细菌过滤器(50 μm,Sysmex)将样品转移到FACS聚苯乙烯管中,并使用S3TM Cell Sorter(BioRad)将巨噬细胞分选到100 μL PBS中。通过荧光显微镜和微分干涉对比验证分离的细胞。

### 基因表达分析

对100,000个分离的巨噬细胞进行基因表达分析。如巨噬细胞分离部分所述,通过细胞分选器(S3e Cell Sorter,BioRad)分离巨噬细胞,转移到TRIzol试剂(Invitrogen),并使用DEPC处理的研杵均质化。随后,根据制造商的方案用TRIzol试剂(Invitrogen)提取RNA。使用由oligo(dT)20引物引发的Superscript III逆转录酶(Invitrogen)进行逆转录。在CFX 1000 Touch实时循环仪(BioRad)上使用TP 2× SYBR Master Mix(Top-Bio)对特定基因的相对表达率进行定量,采用三个技术重复和以下方案:初始变性-95°C 3分钟,扩增-94°C 15秒、56°C 20秒和72°C 25秒,共40个循环。在65–85°C/步0.5°C进行熔解曲线分析。使用双delta Ct分析分析qPCR数据,并将特定基因的表达归一化为相应样品中核糖体蛋白49(Rp49)的表达。图表中显示相对于对照的相对值(倍数变化)。基因表达分析的样品来自三个独立实验。

### 引物序列

Rp49正向:AAGCTGTCGCACAAATGGCG Rp49反向:GCACGTTGTGCACCAGGAAC Hemolectin正向:GCGTACGAAGGAGATTCTC Hemolectin反向:CACCTCGTGCTTCTGTGT Croquemort正向:CTTCTGGCCGGGTATTGCAG Croquemort反向:GCTTTCATAGGCATCAGT 乳酸脱氢酶正向:CAGAGAAGTGGAACGAGCTG 乳酸脱氢酶反向:CATGTTCGCCCAAAACGGAG Basket正向:TACGGCCCATAGGATCAGGT Basket反向:CCCTATATGCTCGCTTGGCA Relish正向:ACAGGACCGCATATCG Relish反向:GTGGGGTATTTCCGGC Diptericin A正向:GCTGCGCAATCGCTTCTACT Diptericin A反向:TGGTGGAGTGGGCTTCATG Defensin正向:GTTCTTCGTTCTCGTGG Defensin反向:CTTTGAACCCCTTGGC Metchnikowin正向:AACTTAATCTTGGAGCGA Metchnikowin反向:CGGTCTTGGTTGGTTAG Drosocin正向:CCATCGTTTTCCTGCT Drosocin反向:CCATCGTTTTCCTGCT 烯醇化酶正向:CAACATCCAGTCCAACAAGG 烯醇化酶反向:GTTCTTGAAGTCCAGATCGT 磷酸果糖激酶正向:AGCTCACATTTCCAAACATCG 磷酸果糖激酶反向:TTTGATCACCAGAATCACTGC 磷酸葡萄糖异构酶正向:ACTGTCAATCTGTCTGTCCA 磷酸葡萄糖异构酶反向:GATAACAGGAGCATTCTTCTCG Unpaired3正向:AGAACACCTGCAATCTGAAGC Unpaired3反向:TCTTGGTGCTCACTGTGGCC Imaginal morphogenesis protein late 2正向:TTCGCGGTTTCTGGGCACCC Imaginal morphogenesis protein late 2反向:GCGCGTCCGATCGTCGCATA Eiger正向:AGCTGATCCCCCTGGTTTTG Eiger反向:GCCAGATCGTTAGTGCGAGA Stat92E正向:CTGGGCATTCACAACAATCCAC Stat92E反向:GTATTGCGCGTAACGAACCG

## 结果与讨论

### mGPs掺入IONs后的物理化学性质

通过喷雾干燥掺入IONs后,mGPs保留了普通GPs特有的褶皱椭球形状(图2a,b)。通过激光衍射确定的mGPs的体积平均粒径为5.1 ± 1.9 μm(图2c),这与原始酵母的大小和先前报道的未修饰GPs的值一致。磁性颗粒的掺入没有引起mGPs的聚集或表面形态的改变,这一事实对于随后被吞噬细胞的摄取至关重要。普通GPs和mGPs的能量色散X射线光谱(EDX)(图2d,e)证明了mGPs中IONs的存在。通过EDX确定的mGPs的Fe含量为1.4%(表1)。通过AAS独立确定的铁含量为1.2 ± 0.1%。TEM分析显示,IONs均匀分布在mGPs的多糖壳内(图2f)。在掺入mGPs之前,葡聚糖包覆的IONs的体积平均直径为124.1 nm(通过DLS在水中测量),多分散性指数为0.144(图2g插图)。掺入mGPs后,IONs在葡聚糖壳内保持良好分散(图2g)。请注意,在TEM图像中可见为较暗斑点的单个氧化铁核心小于通过DLS测量的完全水合的葡聚糖包覆IONs的等效流体动力学直径。这是因为葡聚糖涂层与β-葡聚糖背景无法区分,而且已知磁性纳米颗粒在水性介质中会形成临时簇。

**表1** mGPs样品的EDX分析

| 样品 | 元素符号 | 原子序数 | 原子浓度% | |------|---------|---------|----------| | 普通GPs | C | 6 | 81.7 | | | O | 8 | 18.3 | | | Fe | 26 | 0.0 | | mGPs | C | 6 | 76.9 | | | O | 8 | 21.7 | | | Fe | 26 | 1.4 |

**图2** (a)普通葡聚糖颗粒的SEM。(b)mGPs的SEM。两个SEM中的比例尺均为8 μm。(c)mGPs在水中的粒径分布,通过静态光散射测量;体积平均粒径为5.1 ± 1.9 μm。(d)普通GPs的EDX光谱。(e)mGPs的EDX光谱,证明铁的存在。mGPs中氧化铁的宏观表现是其被磁铁吸引,如插图所示。(f)单个mGP的TEM。比例尺代表1000 nm。(g)详细TEM显示IONs如何被截留并均匀分散在mGP壳内。比例尺代表200 nm。掺入mGPs前葡聚糖包覆IONs在水中的体积加权粒径分布(通过DLS测量)显示为插图。(h)IONs、普通GPs和mGPs的XRPD光谱,证明mGPs中氧化铁的存在。

通过测量XRPD光谱(图2h)进一步证明了复合mGPs中氧化铁的存在。氧化铁在21.5°、35.1°、67.3°和74.4° 2θ处的特征结晶峰在mGPs中清晰可见,而在普通GPs中不存在此类峰。关于进一步应用的一个关键特征是mGPs在水性介质中关于ION保留的稳定性。为了检测在水性介质中磁性操作期间IONs的潜在损失,通过磁铁反复分离mGPs并重新分散。在上清液中未检测到游离的IONs,表明IONs在多糖壳中的嵌入足够强,可以防止磁性随时间的损失。IONs磁性特性的完整表征,包括5和300 K下的磁化曲线以及场冷和零场冷磁化率,已在我们最近的工作中报道。其磁性特性的宏观表现是mGPs被永磁体吸引并从溶液中分离的能力,如图2所示。

### mGPs的生物分布和巨噬细胞摄取

为了研究mGPs的生物分布和随后活体巨噬细胞的磁性分离,使用了在巨噬细胞中携带GFP蛋白内源表达构建体的黑腹果蝇品系(Crq > Gal4;UAS2xGFP)。这种巨噬细胞易于识别,可用于评估其形态和计数。注射0.1% w/w mGPs导致通过果蝇的开放循环系统快速全身分布(图3a)。注射后20–30分钟内,mGPs可分布于成年果蝇的全身,包括远端部分。注射后1小时内,在与巨噬细胞占据区域中可观察到明显的共定位(图3b),这与早期报道的普通GPs的体内行为一致。通过SEM和TEM对全身横截面的分析已证明mGPs被巨噬细胞内化(图3c–e)。对解剖的免疫细胞的分析显示,巨噬细胞内化了多个mGPs(图3f)。在对照实验中,注射到成年果蝇中的游离IONs(未包封在mGPs中)未发现特异性积累在巨噬细胞中(图S1,支持信息)。

**图3** (a)注射后mGP在果蝇中生物分布的时间进程。20分钟内,mGPs到达成年果蝇身体的远端部分。(b)注射后1小时mGPs(红色)在成年果蝇中的分布,显示与巨噬细胞(绿色)的共定位。(c)伪彩色SEM显微照片,显示注射后20分钟巨噬细胞(绿色)吞噬mGPs(红色)的过程。(d)伪彩色TEM显微照片,显示注射后1小时内吞的mGPs(红色)在巨噬细胞(绿色)中的定位。(e)TEM显微照片,显示内吞的mGPs(红色)在果蝇巨噬细胞(绿色)胞质中的细节。(f)注射mGPs(红色)后1小时CrqGal4 > GFP成年果蝇中吞噬细胞(绿色)的代表性共聚焦图像。肌动蛋白用鬼笔环肽(青色)染色。

### 磁细胞分离和基因表达

注射mGPs后45分钟将果蝇均质化,将匀浆用于磁柱分离(QuadroMACS分离器,LS柱,Miltenyi Biotec)。平行地,通过FACS分离表达GFP的巨噬细胞来处理仅注射缓冲液的果蝇的组织匀浆作为对照(图4a)。基于四个独立生物学重复的伴随图4a的统计数据总结在表2中。磁性分离前,匀浆含有0.458% ± 0.049%的GFP阳性细胞(巨噬细胞)。磁性分离后的残留物含有0.042% ± 0.006%的GFP阳性细胞,约占原始细胞的9.3%。因此,磁性分离能够提取匀浆中最初存在的约90.7%的所有GFP阳性细胞,这与从FACS获得的产率相当。该方法的灵敏度(定义为mGP给药靶向的巨噬细胞比例)为97.9% ± 2.5%(N = 90;4个重复),而其选择性(定义为已吞噬mGPs的细胞群体中巨噬细胞的比例)为100% ± 0%(N = 100;5个重复)。灵敏度和选择性测量的详细信息在支持信息中提供。

从两种方法获得的样品中随后分离RNA提供了可比量的RNA(图4d)。这通过定量纳米滴仪器上的纯化RNA和定量Rp49的表达水平得到证实,Rp49通常用作果蝇中的管家基因。通过mGPs和FACS分离的巨噬细胞中Rp49的浓度分别为630.6 ± 117.3和586.9 ± 115.4 ng/μL。

**表2** 伴随图4a的分选数据

| 磁性分离前 | 重复1 | 重复2 | 重复3 | 重复4 | 平均值 | 标准差 | |------------|-------|-------|-------|-------|--------|--------| | 分选细胞 | 10,123,021 | 10,185,447 | 10,066,524 | 10,121,254 | 10,124,062 | 48,606 | | GFP阳性 | 43,528 | 52,561 | 48,211 | 41,231 | 46,383 | 5040 | | 百分比 | 0.430 | 0.516 | 0.479 | 0.407 | 0.458 | 0.049 |

| 磁性分离后 | 重复1 | 重复2 | 重复3 | 重复4 | 平均值 | 标准差 | |------------|-------|-------|-------|-------|--------|--------| | 分选细胞 | 10,185,894 | 10,024,653 | 10,144,874 | 10,132,241 | 10,121,916 | 68,768 | | GFP阳性 | 4086 | 5112 | 3844 | 4117 | 4290 | 562 | | 百分比 | 0.040 | 0.051 | 0.038 | 0.041 | 0.042 | 0.006 |

**图4** (a)细胞分离过程的示意图。上图:向CrqGal4 > GFP成年果蝇注射50 nL 0.1%(w/w)mGPs。将果蝇均质化,将匀浆磁性筛分,保留约90%的吞噬细胞。收集流穿液,根据内源性表达的GFP信号通过FACS分选(G2门)。分选器检测到剩余的10%未分离的巨噬细胞,占总细胞数的0.04%。下图:在没有mGP注射的参考巨噬细胞分离实验中,仅通过FACS从匀浆中分选巨噬细胞,产率为总细胞数的0.46%(表2)。通过mGPs基磁性分离和FACS分选器获得的吞噬细胞显示出相当的活力,随后用于RT-qPCR。(b)成年果蝇注射mGPs的可视化。(c)磁性分离后活巨噬细胞中croquemort和鬼笔环肽的共聚焦显微镜可视化。(d)磁性和FACS分选巨噬细胞中Rp49(通常用作果蝇中的管家基因)表达水平的定量。

通过台盼蓝测定确定的磁性分离巨噬细胞的活力为95.5%。分离细胞的良好状态还表现为它们在显微镜载玻片表面的特征性铺展表型和细胞骨架重塑(图4c)。最后,分析了两种技术的巨噬细胞特异性标志物(hemolectin、croquemort)、免疫相关基因(defensin、drosocin、metchnikowin、diptericin A)和细胞应激途径特征性读数(Relish、basket)的表达水平,结果表明通过磁性葡聚糖颗粒分离的巨噬细胞具有自然的生理特征(图5)。这表明mGPs没有细胞毒性,其摄取未引起巨噬细胞任何异常的生理反应。未发现炎症细胞因子的表达水平在磁性分离和FACS分选的巨噬细胞之间存在显著差异(图5),表明mGPs的吞噬或磁性分离过程本身均未导致炎症反应的激活。通过mGPs分离的巨噬细胞原则上可随后用于各种分析,如基因表达分析、代谢组学、蛋白质组学、单细胞转录组学和酶活性分析。

**图5** 通过mGPs基磁性分离和FACS分选器获得的吞噬细胞中巨噬细胞标志物(croquemort、hemolectin)、糖酵解基因(乳酸脱氢酶、烯醇化酶、磷酸果糖激酶、磷酸葡萄糖异构酶)、应激和免疫反应基因(basket、Relish、STAT92e)、抗菌肽(metchnikowin、diptericin A、drosocin、defensin)和细胞因子(Eiger、Upd2、Upd3、ImpL2)基因表达的比较。结果通过双因素方差分析后进行Tukey多重比较检验进行比较。针对Rp49归一化的表达水平报告为相对于mGPs分离吞噬细胞中分析基因表达水平的倍数变化,其被任意设置为1。单个点代表生物学重复,线/条显示平均值±SD,星号标记统计学显著差异(*p < 0.05;**p < 0.01),NS标记统计学无显著差异。

## 结论

我们使用了一种基于喷雾干燥过程中快速溶剂蒸发期间多孔多糖壳退溶胀的新方法制备了mGPs。这使得大量独立制备的IONs能够不可逆地截留在mGPs结构中,在其中它们保持均匀分散,没有发生不良的聚集或簇集。当注射到活体果蝇中时,mGP迅速遍布全身,并被巨噬细胞快速且选择性地摄取。这使得能够从组织匀浆中通过磁性分离柱实现随后的巨噬细胞分离。mGPs成功应用于磁细胞分离的关键在于三个特性:(i)保留了原始GPs特有的尺寸、表面形态和结构基团,这是免疫识别和高效吞噬的先决条件;(ii)高浓度的嵌入IONs,这是产生颗粒对外部磁场足够强响应的先决条件;(iii)生物相容性,这是分离细胞良好活力和进一步应用的先决条件,且不损害正常细胞功能和基因表达。

与基于通过特异性抗体将磁珠连接到细胞外表面进行磁性分离的方法相比,基于mGPs的方法具有几个优点:(i)能够实现免疫细胞的无抗体和无标记分离;(ii)覆盖宿主生物体中可能参与病原体吞噬的所有细胞,无需事先了解这些细胞;(iii)由于高度进化保守的特征(吞噬作用),该方法基本上可用于所有动物,而不仅仅是昆虫;(iv)该方法允许短处理时间,操作温和,细胞仅暴露于生理缓冲液,无需额外的化学物质。

总体而言,可以得出结论,磁性酵母GPs(mGPs)的制备代表了分离巨噬细胞的合适策略,其数量和质量足以进行基因表达分析。由于这种方法不依赖于内源性表达的荧光标记物或通过针对表面抗原表位的特异性抗体结合细胞,它也可以适用于希望从昆虫和非昆虫物种中分离活体吞噬细胞群体的其他情况。当然,还应注意,巨噬细胞中mGPs的存在可能并非普遍可取(例如,在研究铁代谢时),但基于本工作提供的数据(活力、功能和基因表达),磁性分离的巨噬细胞未受到mGPs吞噬的负面影响。

## 支持信息可用

支持信息可在https://pubs.acs.org/doi/10.1021/acsbiomaterials.3c01199免费获取。游离IONs(即未嵌入mGPs内)注射到果蝇中的参考实验结果;关于磁性分离方法的选择性、灵敏度和纯度评估的信息;以及关于细胞分选所用门控策略的信息(PDF)。

## 作者贡献

G.K.和I.S.对本工作做出了同等贡献。I.S.、G.K.、A.B.和F.Š.构思了该项目。I.S.、G.K.和V.K.进行了实验。A.B.A.开发了纳米颗粒的制备方法并合成了IONs。P.U.在TEM上分析了纳米颗粒和复合颗粒。I.S.、G.K.、A.B.和F.Š.设计实验并分析结果。A.B.和F.Š.监督研究,提供指导和资金。I.S.、G.K.、A.B.和F.Š.撰写了手稿初稿。I.S.和F.Š.在全体作者的输入下撰写了最终手稿。作者声明没有竞争性的财务利益。

## 致谢

我们要感谢捷克科学基金会的财政支持,项目编号19-26127X(F.Š.)和20-14030S(A.B.)。